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CREB inhibitor
CAS No. 1433286-70-4
CREB inhibitor ( CREB inhibitor )
Catalog No. M20071 CAS No. 1433286-70-4
666-15 is a potent and selective CREB inhibitor (IC50: 81 nM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 102 | In Stock |
|
| 10MG | 160 | In Stock |
|
| 25MG | 327 | In Stock |
|
| 50MG | 520 | In Stock |
|
| 100MG | 750 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameCREB inhibitor
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NoteResearch use only not for human use.
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Brief Description666-15 is a potent and selective CREB inhibitor (IC50: 81 nM).
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Description666-15 is a potent and selective CREB inhibitor (IC50: 81 nM).
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SynonymsCREB inhibitor
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PathwayChromatin/Epigenetic
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TargetEpigenetic Reader Domain
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RecptorCREB
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Research Area——
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Indication——
Chemical Information
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CAS Number1433286-70-4
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Formula Weight620.52
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Molecular FormulaC33H31Cl2N3O5
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Purity>98% (HPLC)
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SolubilityDMSO: 60 mg/mL (96.7 mM)
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SMILESCl.NCCCOc1cc2ccccc2cc1C(=O)NCCOc1cc2ccccc2cc1C(=O)Nc1ccc(Cl)cc1O
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Chemical Name3-(3-Aminopropoxy)-N-[2-[[3-[[(4-chloro-2-hydroxyphenyl)amino]carbonyl]-2-naphthalenyl]oxy]ethyl]-2-naphthalenecarboxamide hydrochloride
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Xie F et al. Identification of a Potent Inhibitor of CREB-Mediated Gene Transcription with Efficacious in Vivo Anticancer Activity. J Med Chem. 2015 Jun 25;58(12):5075-87.
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