CREB inhibitor

CAS No. 1433286-70-4

CREB inhibitor ( CREB inhibitor )

Catalog No. M20071 CAS No. 1433286-70-4

666-15 is a potent and selective CREB inhibitor (IC50: 81 nM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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5MG 102 In Stock
10MG 160 In Stock
25MG 327 In Stock
50MG 520 In Stock
100MG 750 In Stock
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Biological Information

  • Product Name
    CREB inhibitor
  • Note
    Research use only not for human use.
  • Brief Description
    666-15 is a potent and selective CREB inhibitor (IC50: 81 nM).
  • Description
    666-15 is a potent and selective CREB inhibitor (IC50: 81 nM).
  • Synonyms
    CREB inhibitor
  • Pathway
    Chromatin/Epigenetic
  • Target
    Epigenetic Reader Domain
  • Recptor
    CREB
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1433286-70-4
  • Formula Weight
    620.52
  • Molecular Formula
    C33H31Cl2N3O5
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: 60 mg/mL (96.7 mM)
  • SMILES
    Cl.NCCCOc1cc2ccccc2cc1C(=O)NCCOc1cc2ccccc2cc1C(=O)Nc1ccc(Cl)cc1O
  • Chemical Name
    3-(3-Aminopropoxy)-N-[2-[[3-[[(4-chloro-2-hydroxyphenyl)amino]carbonyl]-2-naphthalenyl]oxy]ethyl]-2-naphthalenecarboxamide hydrochloride

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Xie F et al. Identification of a Potent Inhibitor of CREB-Mediated Gene Transcription with Efficacious in Vivo Anticancer Activity. J Med Chem. 2015 Jun 25;58(12):5075-87.
molnova catalog
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